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    Clonazolam molecular structure

    Clonazolam Stats & Data

    C-lam Clonitrazolam clam
    NPS DataHub
    MW353.77
    FormulaC17H12ClN5O2
    CAS33887-02-4
    IUPAC6-(2-Chlorophenyl)-1-methyl-8-nitro-4H-s-triazolo(4,3-a)-(1,4)-benzodiazepine
    SMILESO=N(=O)c1ccc2n3c(C)nnc3CN=C(c3ccccc3Cl)c2c1
    InChIKeyXJRGLCAWBRZUFC-UHFFFAOYSA-N
    Benzodiazepines; 2020/3. Benzodiazepine; 2021/3. Benzodiazepine; 2022/3. Benzodiazepine
    Chemical Class Benzodiazepine
    Psychoactive Class Depressant

    Interaction Warnings

    dissociatives

    This combination can result in an increased risk of vomiting during unconsciousness and death from the resulting suffocation. If this occurs, users should attempt to fall asleep in the recovery position or have a friend move them into it.

    stimulants

    It is dangerous to combine benzodiazepines with stimulants due to the risk of excessive intoxication. Stimulants decrease the sedative effect of benzodiazepines, which is the main factor most people consider when determining their level of intoxication. Once the stimulant wears off, the effects of benzodiazepines will be significantly increased, leading to intensified disinhibition as well as other effects.

    Pharmacology

    DrugBank

    Description

    Quahog, unspecified allergenic extract is used in allergenic testing.

    History & Culture

    Clonazolam was first synthesized in 1971 by The Upjohn Company, the pharmaceutical corporation that would later bring alprazolam (Xanax) to market. In the original research, the compound was described as the most active substance in the series of triazolobenzodiazepines tested. Despite this notable potency and coverage by patents, the drug was never developed for clinical use or marketed. The compound remained largely obscure until reports of its use as a research chemical began appearing online around 2013, making it one of the more recently emerged designer benzodiazepines. The European Monitoring Centre for Drugs and Drug Addiction was first notified of clonazolam's presence in the European Union in January 2015, following a report from Sweden. By 2016, detection of novel benzodiazepines had risen markedly across Europe, with over 300,000 tablets containing designer benzodiazepines—including clonazolam, diclazepam, etizolam, and flubromazolam—seized in 2015, nearly double the figure from the previous year. Clonazolam's extreme potency has made it a subject of particular concern within online drug communities. Early forum discussions frequently noted incidents of blackouts and the rapid development of dependence, establishing a reputation that distinguished it from other designer benzodiazepines in circulation. Its microgram-range activity led to distribution methods uncommon for benzodiazepines, with the substance appearing on blotter paper and in volumetrically prepared solutions rather than as raw powder.

    Subjective Effect Notes

    physical: The physical effects of clonazolam can be broken down into several components which progressively intensify proportional to dosage.

    cognitive: The cognitive effects of clonazolam can be broken down into several components which progressively intensify proportional to dosage. The general head space of clonazolam is described by many as one of intense sedation and decreased inhibition. It contains a large number of typical depressant cognitive effects. Paradoxical reactions to benzodiazepines such as increased seizures (in epileptics), aggression, increased anxiety, violent behavior, loss of impulse control, irritability and suicidal behavior sometimes occur (although they are rare in the general population, with an incidence rate below 1%). These paradoxical effects occur with greater frequency in recreational abusers, individuals with mental disorders, children, and patients on high-dosage regimes.

    Effect Profile

    Curated + 28 Reports
    Benzodiazepine 7.6

    Strong anxiolysis, cognitive impairment, and sedation with moderate euphoria

    Anxiolysis×3
    10
    Sedation / Relaxation×2
    84.3
    Motor / Cognitive Impairment×1
    107.7
    Euphoria / Mood Lift×1
    76.4
    Catalog Erowid

    Tolerance & Pharmacokinetics

    drugs.wiki

    Tolerance Decay

    Full tolerance 3d Half tolerance 37d Baseline ~60d

    Cross-Tolerances

    Alprazolam
    85% ●○○
    Diazepam
    85% ●○○
    Clonazepam
    85% ●○○
    Lorazepam
    85% ●○○
    Etizolam
    85% ●○○
    Bromazolam
    85% ●○○
    Flualprazolam
    85% ●○○
    Flubromazolam
    85% ●○○

    Experience Report Analysis

    Erowid
    28 Reports
    2014–2021 Date Range
    28 With Age Data
    14 Effects Detected

    Demographics

    Gender Distribution

    Age Distribution

    Reports Over Time

    Effect Analysis

    Erowid

    Effects aggregated from 28 experience reports (28 Erowid)

    28 Reports
    14 Effects Detected
    7 Positive
    3 Adverse
    4 Neutral

    Effect Sentiment Distribution

    Confidence Distribution

    Positive Effects 7

    Anxiety Suppression 60.7% 70%
    Euphoria 42.9% 70%
    Sedation 28.6% 70%
    Music Enhancement 21.4% 70%
    Empathy 17.9% 70%
    Stimulation 17.9% 70%
    Focus Enhancement 14.3% 70%

    Adverse Effects 3

    Memory Suppression 35.7% 70%
    Confusion 32.1% 70%
    Motor Impairment 14.3% 70%

    Dosage Distribution

    Dose distribution from experience reports

    Median: 0.5 mg IQR: 0.2–1.5 mg n=15

    Real-World Dose Distribution

    62K Doses

    From 63 individual dose entries

    Oral (n=41)

    Median: 0.25mg 25th: 0.2mg 75th: 0.5mg 90th: 0.75mg
    mg/kg median: 0.007 mg/kg 75th: 0.021

    Rectal (n=5)

    Median: 0.05mg 25th: 0.05mg 75th: 0.05mg 90th: 0.05mg

    Sublingual (n=6)

    Median: 0.75mg 25th: 0.31mg 75th: 1.0mg 90th: 2.0mg
    mg/kg median: 0.009 mg/kg 75th: 0.011

    Form / Preparation

    Most common forms and preparations reported

    Body-Weight Dosing

    Dose relative to body weight from reports with weight data

    Median: 0.007 mg/kg IQR: 0.005–0.026 mg/kg n=14

    Redose Patterns

    Redosing behavior across 23 reports

    39.1% Redosed
    1.7 Avg Doses
    20m Median Interval

    Legal Status

    Country Status Notes
    Australia Schedule 9 Classified as a Schedule 9 prohibited substance under federal law. Substances in this category are considered to have no recognized therapeutic value and high potential for misuse.
    Canada Schedule 4 Listed under Schedule 4 of the Controlled Drugs and Substances Act, restricting possession and distribution without authorization.
    Czech Republic Schedule I (List 4) Controlled under § 1, d), 2. of Nařízení vlády č. 463/2013 Sb. Use is restricted exclusively to limited research purposes or very limited therapeutic applications.
    Germany Anlage II BtMG Controlled under the Betäubungsmittelgesetz (Narcotics Act) since November 11, 2021. Production and import with intent to distribute, administration to another person, possession, and trading are prohibited.
    Japan Controlled Regulated under the Pharmaceutical Affairs Law. Possession and sale are illegal without authorization.
    Netherlands List 2 (Opiumwet) Controlled as a List 2 substance under the Opium Law. Possession, production, and distribution are illegal.
    Poland NPS Class Classified as a New Psychoactive Substance under Polish drug legislation. Possession and distribution are prohibited.
    Russia Schedule III Listed as a Schedule III controlled substance since 2017. Subject to restrictions on production, distribution, and possession.
    Sweden Hazardous Substance Classified as an addictive substance following a recommendation by Sweden's public health agency on June 1, 2015. Production, import, trading, and possession require special authorization.
    Switzerland Verzeichnis E Specifically named as a controlled substance under Verzeichnis E (List E) of Swiss narcotics legislation.
    United Kingdom Class C Classified as a Class C drug under the May 2017 amendment to the Misuse of Drugs Act 1971, alongside several other designer benzodiazepines. Possession, production, and supply are criminal offenses.
    United States Schedule I Temporarily placed under Schedule I of the Controlled Substances Act effective July 26, 2023, following DEA consideration announced in December 2022. The temporary scheduling has been extended until July 26, 2026. Not FDA approved for human consumption. Several states enacted their own scheduling prior to federal action, including Virginia, Oregon, and Minnesota (since August 2020).
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