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    EPH molecular structure

    EPH Stats & Data

    Ep Epd Ethylcaine Ethylphenidate
    NPS DataHub
    MW247.34
    FormulaC15H21NO2
    CAS57413-43-1
    IUPACethyl 2-phenyl-2-piperidin-1-ylacetate
    SMILESCCOC(=O)C(N1CCCCC1)c1ccccc1
    InChIKeyAGSKYKDXQOBAPX-UHFFFAOYSA-N
    Piperidines & pyrrolidines
    Chemical Class Phenethylamine
    Psychoactive Class Stimulant

    Interaction Warnings

    mdma

    The neurotoxic effects of MDMA may be increased when combined with other stimulants.

    cocaine

    This combination may increase strain on the heart.

    History & Culture

    Ethylphenidate emerged on the recreational drug market around 2010-2011 and gained increasing popularity over the subsequent years. It became primarily distributed as a research chemical through online vendors, exploiting its grey-area legal status in various jurisdictions during this period. The substance was also stocked by head shops in major cities across the United Kingdom and elsewhere, where it was sometimes sold both as a standalone product and as a component of blended preparations. One notable example was certain formulations marketed as "GoGaine," which combined ethylphenidate with other substances including MPA, lidocaine, and mannitol. An interesting aspect of ethylphenidate's pharmacological history relates to its endogenous formation within the human body. Small quantities of ethylphenidate can be produced through hepatic transesterification when ethanol and methylphenidate are co-ingested. This metabolic pathway parallels the formation of cocaethylene when cocaine and alcohol are consumed together. However, only a small percentage of consumed methylphenidate undergoes this conversion, meaning pharmacologically significant concentrations with measurable physiological effects would not typically be produced through this mechanism under normal circumstances. The phenomenon is most likely to occur in scenarios involving large quantities of both substances, such as in cases of non-medical use or overdose.

    Subjective Effect Notes

    physical: The physical effects of ethylphenidate can be broken down into several components which progressively intensify proportional to dosage.

    cognitive: The cognitive effects of ethylphenidate can be broken down into several components which progressively intensify proportional to dosage. The general head space of ethylphenidate is described by many as one of extreme mental stimulation, increased focus, and powerful euphoria. It contains a large number of typical stimulant cognitive effects. Although negative side effects are usually mild at low to moderate dosages, they become increasingly likely to manifest themselves with higher amounts or extended usage. This particularly holds true during the offset of the experience.

    Effect Profile

    Curated + 51 Reports
    Stimulant 8.8

    Strong stimulation, euphoria, focus, and anxiety/jitters

    Stimulation / Energy×3
    1010
    Euphoria / Mood Lift×2
    1010
    Focus / Productivity×2
    108.2
    Anxiety / Jitters×1
    1010
    Catalog Erowid

    Tolerance & Pharmacokinetics

    drugs.wiki

    Tolerance Decay

    Full tolerance 1h Half tolerance 10d Baseline ~14d

    Experience Report Analysis

    Erowid
    51 Reports
    2011–2018 Date Range
    48 With Age Data
    27 Effects Detected

    Demographics

    Gender Distribution

    Age Distribution

    Reports Over Time

    Effect Analysis

    Erowid

    Effects aggregated from 51 experience reports (51 Erowid)

    51 Reports
    27 Effects Detected
    9 Positive
    11 Adverse
    7 Neutral

    Effect Sentiment Distribution

    Confidence Distribution

    Positive Effects 9

    Euphoria 70.6% 70%
    Stimulation 70.6% 70%
    Focus Enhancement 41.2% 70%
    Music Enhancement 33.3% 70%
    Empathy 31.4% 70%
    Color Enhancement 13.7% 70%
    Introspection 11.8% 70%
    Body High 7.8% 70%
    Tactile Enhancement 7.8% 70%

    Adverse Effects 11

    Anxiety 52.9% 70%
    Jaw Clenching 23.5% 70%
    Increased Heart Rate 23.5% 70%
    Confusion 21.6% 70%
    Sweating 19.6% 70%
    Muscle Tension 13.7% 70%
    Pupil Dilation 11.8% 70%
    Nausea 11.8% 70%
    Appetite Suppression 7.8% 70%
    Motor Impairment 7.8% 70%
    Psychosis 7.8% 70%

    Dose-Response Correlation

    How effect frequency changes across dose levels

    View data table
    Effect Threshold (n=17)
    Stimulation 82.4%
    Euphoria 76.5%
    Anxiety 58.8%
    Music Enhancement 47.1%
    Empathy 41.2%
    Focus Enhancement 41.2%
    Jaw Clenching 35.3%
    Confusion 29.4%
    Color Enhancement 23.5%
    Introspection 17.6%
    Sweating 17.6%
    Pupil Dilation 17.6%
    Sedation 17.6%
    Auditory Effects 17.6%
    Nausea 17.6%

    Dose–Effect Mapping

    Experience Reports

    How reported effects shift across dose tiers, based on 51 experience reports.

    Limited tier coverage — most reports fall within the Threshold range. Effects at other dose levels may not be represented.

    Insufflated dose range: 20.0–50.0 mg (median 25.0 mg)
    Effect Threshold (n=17)
    stimulation
    82%
    euphoria
    76%
    anxiety
    59%
    music enhancement
    47%
    empathy
    41%
    focus enhancement
    41%
    jaw clenching
    35%
    confusion
    29%
    color enhancement
    24%
    introspection
    18%
    sweating
    18%
    pupil dilation
    18%
    sedation
    18%
    auditory effects
    18%
    nausea
    18%
    appetite suppression
    12%
    ego dissolution
    12%
    tactile enhancement
    12%
    increased heart rate
    12%

    Dosage Distribution

    Dose distribution from experience reports

    Median: 25.0 mg IQR: 20.0–50.0 mg n=17

    Real-World Dose Distribution

    62K Doses

    From 113 individual dose entries

    Oral (n=31)

    Median: 15.0mg 25th: 7.0mg 75th: 20.0mg 90th: 50.0mg
    mg/kg median: 0.368 mg/kg 75th: 0.667

    Rectal (n=10)

    Median: 8.0mg 25th: 7.0mg 75th: 9.0mg 90th: 9.0mg

    Insufflated (n=55)

    Median: 25.0mg 25th: 17.5mg 75th: 50.0mg 90th: 50.0mg
    mg/kg median: 0.333 mg/kg 75th: 0.589

    Form / Preparation

    Most common forms and preparations reported

    Body-Weight Dosing

    Dose relative to body weight from reports with weight data

    Insufflated

    Median: 0.333 mg/kg IQR: 0.275–0.59 mg/kg n=15

    Oral

    Median: 0.5 mg/kg IQR: 0.275–0.667 mg/kg n=6

    Redose Patterns

    Redosing behavior across 49 reports

    49.0% Redosed
    2.2 Avg Doses
    60m Median Interval

    Legal Status

    Not controlled under international drug treaties
    Country Status Notes
    Australia Controlled (analogue provisions) Australian state and federal legislation contains provisions covering analogues of controlled drugs. Ethylphenidate falls under these provisions as an analogue of methylphenidate.
    Austria Illegal (NPSG) Prohibited since January 1, 2012 under the Neue-Psychoaktive-Substanzen-Gesetz (New Psychoactive Substances Act).
    Canada Schedule III (CDSA) Listed on the Controlled Drugs and Substances Act in Schedule III as of May 5, 2017. Previously unscheduled with no analog law covering it.
    Denmark Illegal Controlled substance as of February 1, 2013.
    Germany Anlage II BtMG Controlled under Anlage II of the Betäubungsmittelgesetz (Narcotics Act) as of July 17, 2013. Manufacturing, possession, import, export, purchase, sale, procurement, and dispensing without a license is prohibited.
    Jersey Illegal Controlled under the Misuse of Drugs (Jersey) Law 1978.
    Netherlands Lijst I (Opiumwet) Listed in Lijst I of the Opiumwet (Opium Act) as of April 27, 2018.
    Norway Unscheduled Not specifically listed as controlled under the Forskrift om narkotika (narcotics regulation). Despite structural similarity to methylphenidate, Norwegian law does not automatically control ethylphenidate as an analogue.
    Sweden Illegal (Appendix 1) Listed in Appendix 1 of Swedish drug control regulations as of December 15, 2012, making it illegal for most purposes.
    Switzerland Controlled (Verzeichnis D) Specifically named as a controlled substance under Verzeichnis D of Swiss drug regulations.
    United Kingdom Class B Initially placed under emergency control as a Temporary Class Drug in April 2015 along with other phenidates, restricting sale and manufacture. Subsequently classified as a Class B drug on May 31, 2017, making possession, production, and supply illegal.
    United States Unscheduled (federally) Not explicitly scheduled at the federal level. However, as a structural analogue of methylphenidate (Schedule II), it could potentially be prosecuted under the Federal Analogue Act if sold for human consumption or possessed with intent to ingest. Specifically controlled in Utah along with its analogues, homologs, and synthetic equivalents.
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