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    Methamphetamine molecular structure

    Methamphetamine Stats & Data

    meth desoxyn tik
    NPS DataHub
    MW149.24
    FormulaC10H15N
    CAS537-46-2
    IUPAC~{N}-methyl-1-phenylpropan-2-amine
    SMILESCNC(C)Cc1ccccc1
    InChIKeyMYWUZJCMWCOHBA-UHFFFAOYSA-N
    Phenethylamines; 2020/1. Von 2-Phenethylamin abgeleitete Verbindungen; 2021/1. Von 2-Phenethylamin abgeleitete Verbindungen; 2022/1. Von 2-Phenethylamin abgeleitete Verbindungen
    Chemical Class Amphetamine
    Psychoactive Class Stimulant
    Half-Life Highly variable; typical ≈ 9–12 h, strongly influenced by urine pH (reports range from ~4–5 h to >20 h).

    Interaction Warnings

    tricyclic antidepressants

    Amphetamine may increase the effects of tricyclic antidepressants to dangerous levels.

    mdma

    The neurotoxic effects of MDMA may be increased when combined with amphetamines.

    cocaine

    This combination may increase strain on the heart.

    Pharmacology

    DrugBank
    State Solid

    Description

    Metamfetamine (methamphetamine) is a psychostimulant and sympathomimetic drug. It is a member of the amphetamine group of sympathomimetic amines. Methamphetamine can induce effects such as euphoria, increased alertness and energy, and enhanced self-esteem. It is a scheduled drug in most countries due to its high potential for addiction and abuse.

    Mechanism of Action

    Methamphetamine enters the brain and triggers a cascading release of norepinephrine, dopamine and serotonin. To a lesser extent methamphetamine acts as a dopaminergic and adrenergic reuptake inhibitor and in high concentrations as a monamine oxidase inhibitor (MAOI). The mechanism of action involved in producing the beneficial behavioral changes seen in hyperkinetic children receiving methamphetamine is unknown.

    Pharmacodynamics

    Methamphetamine is a potent central nervous system stimulant which affects neurochemical mechanisms responsible for regulating heart rate, body temperature, blood pressure, appetite, attention, mood and responses associated with alertness or alarm conditions. The acute effects of the drug closely resemble the physiological and psychological effects of an epinephrine-provoked fight-or-flight response, including increased heart rate and blood pressure, vasoconstriction (constriction of the arterial walls), bronchodilation, and hyperglycemia (increased blood sugar). Users experience an increase in focus, increased mental alertness, and the elimination of fatigue, as well as a decrease in appetite.

    Metabolism

    Hepatic. The primary site of metabolism is in the liver by aromatic hydroxylation, N-dealkylation and deamination. At least seven metabolites have been identified in the urine, with the main metabolites being amphetamine (active) and 4-hydroxymethamphetamine. Other minor metabolites include 4-hydroxyamphetamine, norephedrine, and 4-hydroxynorephedrine.

    Absorption

    Methamphetamine is rapidly absorbed from the gastrointestinal tract with peak methamphetamine concentrations occurring in 3.13 to 6.3 hours post ingestion. Moreover, when administered intranasally or as an inhalation, methamphetamine also demonstrates a high degree of absorption. It is distributed to most parts of the body. Because methamphetamine has a high lipophilicity it is distributed across the blood brain barrier and crosses the placenta.

    Toxicity

    Manifestations of acute overdosage with methamphetamine include restlessness, tremor, hyperreflexia, rapid respiration, confusion, assaultiveness, hallucinations, panic states, hyperpyrexia, and rhabdomyolysis. Fatigue and depression usually follow the central stimulation. Cardiovascular effects include arrhythmias, hypertension or hypotension, and circulatory collapse. Gastrointestinal symptoms include nausea, vomiting, diarrhea, and abdominal cramps. Fatal poisoning usually terminates in convulsions and coma.

    Indication

    For the treatment of Attention Deficit Disorder with Hyperactivity (ADHD) and exogenous obesity.

    Half-life

    The biological half-life has been reported in the range of 4 to 5 hours.

    Elimination

    Excretion occurs primarily in the urine, the rate of which is dependent on urine pH. Between 30-54% of an oral dose is excreted in urine as unchanged methamphetamine and 10-23% as unchanged amphetamine. Following an intravenous dose, 45% is excreted as unchanged parent drug and 7% amphetamine.

    Receptor Profile

    Receptor Actions

    Inhibitors
    Dopamine reuptake inhibitor
    Norepinephrine reuptake inhibitor
    Monoamine oxidase inhibitor (high concentrations)
    Other
    Dopamine releasing agent
    Norepinephrine releasing agent
    Serotonin releasing agent

    History & Culture

    1893–1919

    The development of methamphetamine followed shortly after the creation of its parent compound. Romanian chemist Lazăr Edeleanu first synthesized amphetamine in Germany in 1887, naming it phenylisopropylamine. Six years later, Japanese chemist Nagai Nagayoshi achieved the first synthesis of methamphetamine from ephedrine in 1893. Despite these discoveries, neither substance found pharmacological application for several decades. A significant advancement came in 1919 when Japanese pharmacologist Akira Ogata developed a method to produce methamphetamine hydrochloride through the reduction of ephedrine using red phosphorus and iodine. This crystalline salt form would eventually become the basis for both pharmaceutical manufacturing and illicit production.

    1938–1945

    Beginning in 1938, methamphetamine became available as a nonprescription drug in Germany under the brand name Pervitin, manufactured by the Berlin-based Temmler pharmaceutical company. The German military subsequently incorporated the drug across all branches of the armed forces, valuing its stimulant properties and capacity to sustain wakefulness during extended operations. Soldiers gave the tablets colloquial nicknames including "Stuka-Tablets" and "Hermann-Göring-Pills," the latter a sardonic allusion to the Reichsmarschall's well-known drug dependencies. The severe consequences of use, particularly debilitating withdrawal symptoms, prompted military authorities to sharply reduce distribution by 1940. By 1941, access required a prescription, and supply was tightly controlled. Soldiers subsequently received only a few tablets at a time and were discouraged from combat use. As historian Łukasz Kamieński documented, soldiers who took Pervitin before battle typically found themselves unable to function effectively for one to two days afterward, experiencing severe drug hangovers that rendered them ineffective. In some cases, soldiers under the influence committed violent acts against civilians or turned on their own officers. Near the war's conclusion, methamphetamine became a component in an experimental combination drug designated D-IX. Beyond Germany, both Allied and Axis forces employed amphetamines and methamphetamine throughout the conflict for their performance-enhancing and fatigue-reducing properties.

    1950s–1960s

    Following World War II, pharmaceutical methamphetamine transitioned into civilian medical use. Obetrol Pharmaceuticals patented Obetrol in the 1950s, establishing one of the first branded pharmaceutical methamphetamine products indicated for obesity treatment. The drug's psychological and stimulant properties made it an extremely popular weight-loss medication in the United States throughout the 1950s and 1960s. As evidence of the drug's addictive properties accumulated, governments began implementing increasingly strict controls on its production and distribution. Pharmaceutical methamphetamine continues to be marketed under the trade name Desoxyn, with the trademark passing from Lundbeck to Italian pharmaceutical company Recordati in January 2013.

    Illicit methamphetamine production has become concentrated in the Golden Triangle of Southeast Asia, with Shan State in Myanmar emerging as the world's leading manufacturing center. Operations in this region produce both ya ba (the tablet form popular in East Asia) and crystalline methamphetamine for distribution across East and Southeast Asia, the Pacific, and the United States. The Cantonese Chinese syndicate known as Sam Gor, or "The Company," is understood to be the primary international criminal organization driving this production expansion. Comprised of members from five different triads, the organization allegedly controls approximately 40 percent of the Asia-Pacific methamphetamine market while also trafficking heroin and ketamine. Sam Gor generates an estimated minimum of eight billion dollars annually and maintains operations spanning Myanmar, Thailand, New Zealand, Australia, Japan, China, and Taiwan. Previously operating manufacturing facilities in Southern China, the organization relocated production primarily to Shan State, contributing to a massive surge in regional crystal methamphetamine supply around 2019. Despite well-documented risks of dependence and substantial media attention devoted to its dangers, methamphetamine remains widely used as a recreational substance globally.

    Subjective Effect Notes

    physical: The physical effects of Methamphetamine can be broken down into several components which progressively intensify proportional to dosage.

    cognitive: The cognitive effects of methamphetamine can be broken down into several components which progressively intensify proportional to dosage. The general head space of methamphetamine is described by many as one of extreme mental stimulation, increased focus, and powerful euphoria. It contains a large number of typical stimulant cognitive effects. Although negative side effects are usually mild at low to moderate dosages, they become increasingly likely to manifest themselves with higher amounts or extended usage. This particularly holds true during the offset of the experience.

    Effect Profile

    Curated + 711 Reports
    Stimulant 8.4

    Strong stimulation, euphoria, and focus with moderate anxiety/jitters

    Stimulation / Energy×3
    108.6 4/20
    Euphoria / Mood Lift×2
    95.1 18/20
    Focus / Productivity×2
    83.4 3/20
    Anxiety / Jitters×1
    710 4/20
    Catalog Erowid

    User Experiences

    Stimulation "The effect of that tiny bit was so intense I couldn't sleep for 3 days (I lay there at night eyes closed for 8+ hours strait, 2 nights in a row, totally awake, mind flying like crazy trying to sleep)." Bluelight
    Euphoria "If you have a decent size shot of good quality meth that is diluted half water half dope you will prolly get an amazing rush." Bluelight
    Focus "so anyways today i went to buy some, and instead of doing the whole bag of 20 dollars worth like i always do, for someone with no tolerance its too much, and doesn't make you feel anymore amazing..." Bluelight

    Duration Timeline

    Bluelight
    Onset Comeup Peak Offset After Effects
    Smoked
    0-1 minutes
    0-0 minutes
    3.0-8.0 hours
    1-3 hours
    24.0 hours
    Total: 1-3 hours
    Oral
    19 minutes - 1.17 hours
    1-3 hours
    10.0-12.0 hours
    3-4 hours
    24.0 hours
    Total: 3-5 hours
    Insufflated
    4-10 minutes
    3-4 minutes
    8.0-10.0 hours
    2-4 hours
    24.0 hours
    Total: 1-3 hours
    Rectal
    4-15 minutes
    3-4 minutes
    2-4 hours
    3-5 hours
    12-24 hours
    Intravenous
    0-1 minutes
    1-1 minutes
    4.0-8.0 hours
    3-4 hours
    24.0 hours
    Total: 4-8 hours

    Community Effects

    TripSit
    Positive
    euphoria visual enhancement energy
    Negative
    nausea vomiting anxiety paranoia insomnia confusion psychosis addiction

    Tolerance & Pharmacokinetics

    drugs.wiki
    Half-Life
    Highly variable; typical ≈ 9–12 h, strongly influenced by urine pH (reports range from ~4–5 h to >20 h).
    Addiction Potential
    High. Methamphetamine is highly addictive with significant risk of psychological and physical dependence.

    Tolerance Decay

    Full tolerance 2d Half tolerance 14d Baseline ~30d

    Acute tolerance builds rapidly over one or more long sessions, with noticeable blunting on subsequent doses; partial reversal occurs over 1–4 weeks if abstinent. Data are largely observational/anecdotal from user communities rather than controlled studies.

    Cross-Tolerances

    Amphetamine/dextroamphetamine
    50% ●○○

    Experience Report Analysis

    Erowid BlueLight
    560 Reports
    1992–2025 Date Range
    108 With Age Data
    31 Effects Detected

    Demographics

    Gender Distribution

    Age Distribution

    Reports Over Time

    Effect Analysis

    Erowid + Bluelight

    Effects aggregated from 610 experience reports (560 Erowid + 151 Bluelight)

    610 Reports
    139 Effects Detected
    43 Positive
    79 Adverse
    17 Neutral

    Effect Sentiment Distribution

    Confidence Distribution

    Positive Effects 43

    Stimulation 50.5% 86%
    Thought Acceleration 44.0% 81%
    Euphoria 35.0% 90%
    Sociability Enhancement 28.0% 86%
    Empathy 24.7% 82%
    Tactile Enhancement 21.0% 88%
    Focus Enhancement 17.2% 86%
    Music Enhancement 15.6% 80%
    Emotional Openness 12.0% 85%
    Color Enhancement 11.0% 82%
    Body High 10.1% 81%
    Libido Enhancement 10.0% 81%
    Love 8.0% 91%
    Contentment 8.0% 78%
    Motor Enhancement 8.0% 83%
    Empathogenic Connection 8.0% 84%
    Insight 6.0% 79%
    Brightness Enhancement 6.0% 83%
    Peace 6.0% 84%
    Awe 6.0% 80%

    Adverse Effects 79

    Insomnia 50.0% 87%
    Anxiety 45.4% 80%
    Body Load 38.0% 77%
    Confusion 28.8% 80%
    Delusion 20.0% 87%
    Paranoid Ideation 20.0% 89%
    Dry Mouth 20.0% 81%
    Body Temperature Change 18.0% 82%
    Panic 18.0% 85%
    Fear 18.0% 87%
    Tingling 18.0% 87%
    Paranoia 16.0% 87%
    Tremor 12.0% 79%
    Dysphoria 12.0% 81%
    Depersonalization 12.0% 76%
    Nausea 11.2% 85%
    Restlessness 10.0% 76%
    Dizziness 10.0% 83%
    Entity Imagery 10.0% 83%
    Jaw Clenching 8.5% 83%

    Dose-Response Correlation

    How effect frequency changes across dose levels

    Smoked

    View data table
    Effect Heavy (n=23)
    Anxiety 56.5%
    Confusion 56.5%
    Stimulation 56.5%
    Euphoria 30.4%
    Sedation 21.7%
    Psychosis 17.4%
    Color Enhancement 17.4%
    Visual Distortions 13.0%
    Empathy 13.0%
    Tactile Enhancement 13.0%
    Memory Suppression 8.7%
    Hospital 8.7%
    Time Distortion 8.7%
    Dissociation 8.7%
    Increased Heart Rate 8.7%

    Insufflated

    View data table
    Effect Heavy (n=15)
    Stimulation 60.0%
    Anxiety 53.3%
    Euphoria 46.7%
    Sedation 46.7%
    Focus Enhancement 33.3%
    Music Enhancement 26.7%
    Tactile Enhancement 26.7%
    Confusion 20.0%
    Visual Distortions 20.0%
    Color Enhancement 20.0%
    Body High 20.0%
    Auditory Effects 20.0%
    Open-Eye Visuals 20.0%
    Memory Suppression 20.0%
    Increased Heart Rate 20.0%

    Subjective Effect Ontology

    Experience Reports

    Structured effect tags extracted from 711 Erowid & Bluelight experience reports using a controlled vocabulary of 220+ canonical effects across 15 domains.

    Cognitive

    confusion 176 25.9% focus enhancement 105 17.3%

    Emotional

    anxiety 277 43.8% euphoria 213 36.8% empathy 151 22.3%

    Motor

    stimulation 308 53.3% sedation 123 17.6%

    Tactile

    tactile enhancement 128 18.6%

    8 unique effects extracted · Derived from Erowid & Bluelight reports

    Dose–Effect Mapping

    Experience Reports

    How reported effects shift across dose tiers, based on 560 experience reports.

    Limited tier coverage — most reports fall within the Heavy range. Effects at other dose levels may not be represented.

    Insufflated dose range: 65.0–500.0 mg (median 200.0 mg)
    Effect Heavy (n=15)
    stimulation
    60%
    anxiety
    53%
    euphoria
    47%
    sedation
    47%
    focus enhancement
    33%
    music enhancement
    27%
    tactile enhancement
    27%
    confusion
    20%
    visual distortions
    20%
    color enhancement
    20%
    body high
    20%
    auditory effects
    20%
    open-eye visuals
    20%
    memory suppression
    20%
    increased heart rate
    20%
    headache
    13%
    closed-eye visuals
    13%
    sweating
    13%
    appetite suppression
    13%
    empathy
    13%

    Showing top 20 of 21 effects

    Smoked dose range: 300.0–1500.0 mg (median 600.0 mg)
    Effect Heavy (n=23)
    anxiety
    56%
    confusion
    56%
    stimulation
    56%
    euphoria
    30%
    sedation
    22%
    psychosis
    17%
    color enhancement
    17%
    visual distortions
    13%
    empathy
    13%
    tactile enhancement
    13%
    memory suppression
    9%
    hospital
    9%
    time distortion
    9%
    dissociation
    9%
    increased heart rate
    9%

    Dosage Distribution

    Dose distribution from experience reports

    Smoked

    Median: 600.0 mg IQR: 300.0–1500.0 mg n=16

    Oral

    Median: 50.0 mg IQR: 20.0–125.0 mg n=11

    Insufflated

    Median: 200.0 mg IQR: 65.0–500.0 mg n=21

    Real-World Dose Distribution

    62K Doses

    From 919 individual dose entries

    Rectal (n=589)

    Median: 10.0mg 25th: 5.0mg 75th: 20.0mg 90th: 33.0mg

    Oral (n=93)

    Median: 15.0mg 25th: 10.0mg 75th: 20.0mg 90th: 30.0mg
    mg/kg median: 0.825 mg/kg 75th: 2.02

    Smoked (n=27)

    Median: 250.0mg 25th: 100.0mg 75th: 550.0mg 90th: 1200.0mg
    mg/kg median: 3.674 mg/kg 75th: 9.285

    Insufflated (n=37)

    Median: 150.0mg 25th: 30.0mg 75th: 300.0mg 90th: 500.0mg
    mg/kg median: 2.212 mg/kg 75th: 4.674

    Intravenous (n=15)

    Median: 164.0mg 25th: 95.0mg 75th: 250.0mg 90th: 410.0mg
    mg/kg median: 2.92 mg/kg 75th: 3.937

    Common Combinations

    Most co-occurring substances in experience reports

    Form / Preparation

    Most common forms and preparations reported

    Body-Weight Dosing

    Dose relative to body weight from reports with weight data

    Smoked

    Median: 9.119 mg/kg IQR: 1.575–20.661 mg/kg n=15

    Oral

    Median: 1.002 mg/kg IQR: 0.333–2.174 mg/kg n=10

    Intravenous

    Median: 2.051 mg/kg IQR: 0.63–3.082 mg/kg n=5

    Unknown

    Median: 11.811 mg/kg IQR: 7.348–38.911 mg/kg n=10

    Insufflated

    Median: 3.04 mg/kg IQR: 0.724–6.196 mg/kg n=21

    Redose Patterns

    Redosing behavior across 405 reports

    16.8% Redosed
    1.2 Avg Doses
    180m Median Interval

    Legal Status

    UN Convention on Psychotropic Substances 1971 (Schedule II)
    Country Status Notes
    Australia Schedule 8 Available for medical use under Schedule 8, but possession, production, or supply without authority is illegal. Personal quantities under 1.5 grams were decriminalized in the Australian Capital Territory as of October 28, 2023.
    Austria Illegal (SMG) Prohibited under the Suchtmittelgesetz (SMG - Austrian Narcotics Act). Illegal to possess, produce, or sell.
    Brazil Class F2 Listed as a Class F2 prohibited psychoactive substance. Reports indicate it may sometimes be obtained with a prescription.
    Canada Schedule I (CDSA) Listed under Schedule I of the Controlled Drugs and Substances Act since August 2005. Previously classified as Schedule III. A 2011 Supreme Court decision established a constitutional right to access supervised injection sites under Section 7 of the Charter.
    Czech Republic Schedule II Controlled as a Schedule II substance under national drug legislation.
    France Stupéfiant Scheduled as a stupéfiant, a recognized drug of abuse under French law. Illegal to possess, buy, sell, or manufacture.
    Germany Anlage II BtMG First added to the Opiumgesetz (Opium Act) on July 1, 1941. Currently controlled under Anlage II of the Betäubungsmittelgesetz (Narcotics Act) since March 1, 2008. Previously listed in Anlage III, which permitted prescription on narcotic prescription forms. Manufacturing, possession, import, export, purchase, sale, procurement, or dispensing without a license is prohibited.
    Israel Prohibited Banned in July 2010 as part of legislation targeting four families of substances (cathinones, methcathinones, amphetamines, and methamphetamines) along with their derivatives. The framework was designed to preemptively prohibit novel analogues.
    Japan Prohibited Controlled under the Amphetamines Control Law of 1954. Production, distribution, and possession are illegal.
    Netherlands List I (Opiumwet) Controlled as a List I substance under the Opium Act. Possession, distribution, and production without license is illegal.
    New Zealand Class A Controlled as a Class A substance, representing the most restrictive category under New Zealand's drug scheduling system.
    Norway Schedule II Classified as Schedule II under Norwegian drug legislation. Illegal to buy or possess without a prescription.
    Poland Group II-P Controlled as a Group II-P substance under Polish drug legislation.
    South Korea Prohibited Banned in compliance with the United Nations Convention on Psychotropic Substances.
    Sweden List II / List P II Classified under both the 1971 UN Psychotropic Convention (List P II) and domestically under Sweden's List II. Possession, distribution, and production are prohibited.
    Switzerland Verzeichnis A Specifically named as a controlled substance under Verzeichnis A (Schedule A) of Swiss narcotics legislation.
    United Kingdom Class A Classified as Class A, the most restrictive category, since January 18, 2007. Illegal to buy, sell, or possess.
    United States Schedule II Controlled under the Controlled Substances Act since 1970. Available by prescription under the trade name Desoxyn for treatment of ADHD and severe obesity, though rarely prescribed due to abuse potential. Illegal to buy, sell, or possess without a DEA license or prescription. Notably, levomethamphetamine remains available over-the-counter.

    Harm Reduction

    drugs.wiki

    - Purity/formulation matter: street meth is almost always the hydrochloride (HCl) salt, which is water-soluble and directly smokable; meth freebase is an oily liquid and uncommon. Do not attempt to base or re-base street crystals; this creates caustic products and adds risks. Salt-to-base potency differs by ~20% (HCl MW ~185.7 vs base 149.2).

    - Half-life and duration vary with urine pH: alkalinization markedly slows renal clearance and can extend both duration and adverse effects; acidification speeds clearance. Intentionally altering body pH to tweak duration is risky and discouraged.

    - Cardiovascular strain (tachycardia, hypertension, arrhythmia, chest pain) and hyperthermia are leading acute harms; risk escalates with dose, redosing, dehydration, heat, and polydrug stimulant use. Seek urgent care for chest pain, severe headache, or high fever.

    - Neurotoxicity risk increases with high doses, hyperthermia, and prolonged wakefulness; spacing sessions, sleeping, eating, and keeping cool are protective behaviors.

    - Redosing drives binges and insomnia. Plan a cutoff time; dose early in the day; avoid stacking routes (e.g., smoking then IV).

    - Hydration: sip ~250–500 mL/h of water or oral rehydration solution when active/hot; avoid overhydration. Replace electrolytes on long sessions.

    - Oral care: dry mouth (xerostomia) and bruxism increase caries risk. Prefer water over sugary sodas; use sugar-free gum/lozenges for saliva; brush gently before bed; consider fluoride rinse.

    - Insufflation: rotate nostrils; use fine powder; rinse with sterile saline after to reduce irritation and septal damage.

    - Smoking: use heat-control (no direct flame on crystal), avoid sharing pipes/mouthpieces to reduce infection transmission from burns/sores; allow glass to cool to prevent cracks and cuts.

    - Injection: use new sterile equipment every time; filter with a 0.22 μm wheel filter if possible; avoid ‘acidifying’ crystal HCl; rotate sites; never share equipment; watch for signs of infection or endocarditis (fever, chills, new heart murmur).

    - Drug checking: if available, use reagent testing or mail-in lab services. Fentanyl test strips can detect contamination but require high dilution to avoid false positives from concentrated stimulants; test every new batch and carry naloxone where contamination is prevalent.

    - Medicines/supplements: CYP2D6 inhibition (e.g., some antidepressants) can increase active levels; combining with serotonergic or seizure-threshold–lowering drugs (e.g., tramadol) increases risks.

    - Legal status: Schedule II (US) for limited medical uses; illicit supply varies in purity and may include adulterants; never assume any batch is pure.

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