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    4-AcO-DET molecular structure

    4-AcO-DET Stats & Data

    Ethacetin Ethylacybin 4-acetoxy-det
    NPS DataHub
    MW274.36
    FormulaC16H22N2O2
    CAS1135424-15-5
    IUPAC[3-(2-diethylaminoethyl)-1H-indol-4-yl] acetate
    SMILESCCN(CC)CCc1cnc2cccc(OC(C)=O)c12
    InChIKeyWYEVVQJLTXBMPM-UHFFFAOYSA-N
    Tryptamines; 2020/5.1 Indol-3-alkylamine; 2021/5.1 Indol-3-alkylamine; 2022/5.1 Indol-3-alkylamine
    Chemical Class Tryptamine
    Psychoactive Class Psychedelic
    Half-Life Unknown in humans; effects typically persist hours despite rapid onset (likely active metabolite 4-HO-DET).

    Receptor Profile

    Receptor Actions

    Agonists
    5-HT2A receptor agonist (partial)
    Other
    Prodrug (metabolizes to 4-HO-DET)

    History & Culture

    4-AcO-DET was first synthesized in 1958 by Albert Hofmann at the Sandoz laboratories in Switzerland. Despite this early synthesis, the compound remained largely unexplored for decades and has accumulated very little documented history of human usage. In the contemporary era, 4-AcO-DET has found limited use as both a recreational designer drug and an entheogenic compound, with most users acquiring it through online research chemical vendors. It remains relatively rare compared to more widely documented psychedelics in the tryptamine class.

    Effect Profile

    Curated + 50 Reports
    Psychedelic 8.8

    Strong visuals, headspace, auditory effects, and body load

    Visual Intensity×3
    1010
    Headspace Depth×3
    109.4
    Auditory Effects×1
    1010
    Body Load / Somatic Effects×1
    1010
    Catalog Erowid

    Duration Timeline

    Bluelight
    Onset Comeup Peak Offset After Effects
    Oral
    19 minutes - 1.0 hours
    1-1.5 hours
    1.5-3 hours
    1-2 hours
    2-4 hours
    Smoked
    0 minutes
    4-10 minutes
    10-19 minutes
    19-40 minutes
    30 minutes - 1.0 hours

    Tolerance & Pharmacokinetics

    drugs.wiki
    Half-Life
    Unknown in humans; effects typically persist hours despite rapid onset (likely active metabolite 4-HO-DET).
    Addiction Potential
    Not habit-forming; low abuse potential typical of classical psychedelics. Psychological habituation is possible with frequent use.

    Tolerance Decay

    Full tolerance 6h Half tolerance 3d Baseline ~14d

    Estimates inferred from classical psychedelic patterns (psilocybin/LSD) and user reports; quality anecdotal. Avoid redosing to chase effects during the same session due to tolerance spikes and unpredictability.

    Cross-Tolerances

    Psilocybin/Psilocin (4-HO-DMT)
    60% ●○○
    LSD
    50% ●○○
    Other 4-substituted tryptamines (e.g., 4-HO/4-AcO-MET/MiPT)
    60% ●○○

    Experience Report Analysis

    Erowid
    50 Reports
    2001–2021 Date Range
    12 With Age Data
    27 Effects Detected

    Demographics

    Gender Distribution

    Age Distribution

    Reports Over Time

    Effect Analysis

    Erowid

    Effects aggregated from 50 experience reports (50 Erowid)

    50 Reports
    27 Effects Detected
    10 Positive
    9 Adverse
    8 Neutral

    Effect Sentiment Distribution

    Confidence Distribution

    Positive Effects 10

    Music Enhancement 52.0% 70%
    Color Enhancement 50.0% 70%
    Stimulation 46.0% 70%
    Tactile Enhancement 44.0% 70%
    Empathy 42.0% 70%
    Introspection 32.0% 70%
    Euphoria 32.0% 70%
    Focus Enhancement 20.0% 70%
    Body High 18.0% 70%
    Creativity Enhancement 6.0% 70%

    Adverse Effects 9

    Anxiety 48.0% 70%
    Nausea 32.0% 70%
    Muscle Tension 30.0% 70%
    Confusion 28.0% 70%
    Jaw Clenching 14.0% 70%
    Pupil Dilation 8.0% 70%
    Sweating 6.0% 70%
    Increased Heart Rate 6.0% 70%
    Motor Impairment 6.0% 70%

    Dose-Response Correlation

    How effect frequency changes across dose levels

    View data table
    Effect Strong (n=13)
    Visual Distortions 84.6%
    Music Enhancement 53.8%
    Stimulation 46.2%
    Sedation 46.2%
    Color Enhancement 38.5%
    Nausea 38.5%
    Anxiety 38.5%
    Introspection 30.8%
    Muscle Tension 30.8%
    Tactile Enhancement 30.8%
    Focus Enhancement 30.8%
    Confusion 30.8%
    Empathy 23.1%
    Auditory Effects 23.1%
    Open-Eye Visuals 23.1%

    Dose–Effect Mapping

    Experience Reports

    How reported effects shift across dose tiers, based on 50 experience reports.

    Limited tier coverage — most reports fall within the Strong range. Effects at other dose levels may not be represented.

    Oral dose range: 15.0–25.0 mg (median 20.0 mg)
    Effect Strong (n=13)
    visual distortions
    85%
    music enhancement
    54%
    stimulation
    46%
    sedation
    46%
    color enhancement
    38%
    nausea
    38%
    anxiety
    38%
    introspection
    31%
    muscle tension
    31%
    tactile enhancement
    31%
    focus enhancement
    31%
    confusion
    31%
    empathy
    23%
    auditory effects
    23%
    open-eye visuals
    23%
    closed-eye visuals
    15%
    jaw clenching
    15%
    pupil dilation
    15%

    Dosage Distribution

    Dose distribution from experience reports

    Median: 20.0 mg IQR: 15.0–25.0 mg n=27

    Real-World Dose Distribution

    62K Doses

    From 75 individual dose entries

    Oral (n=60)

    Median: 16.0mg 25th: 10.0mg 75th: 20.0mg 90th: 25.5mg
    mg/kg median: 0.252 mg/kg 75th: 0.342

    Insufflated (n=6)

    Median: 17.5mg 25th: 15.0mg 75th: 20.0mg 90th: 27.5mg
    mg/kg median: 0.261 mg/kg 75th: 0.327

    Form / Preparation

    Most common forms and preparations reported

    Body-Weight Dosing

    Dose relative to body weight from reports with weight data

    Median: 0.282 mg/kg IQR: 0.235–0.353 mg/kg n=21

    Redose Patterns

    Redosing behavior across 39 reports

    17.9% Redosed
    1.3 Avg Doses

    Legal Status

    Country Status Notes
    Germany Anlage I BtMG Controlled under Anlage I of the Betäubungsmittelgesetz (Narcotics Act) since January 24, 1974, as it is classified as an ester of DET. Manufacturing, possession, importation, exportation, purchase, sale, and distribution are prohibited without a license.
    Japan Controlled Designated as a controlled substance effective July 29, 2015, under national drug control legislation.
    Sweden Controlled Classified as a health hazard under Lagen om förbud mot vissa hälsofarliga varor (Act on the Prohibition of Certain Goods Dangerous to Health) effective November 1, 2005, under regulation SFS 2005:733. Possession and sale are illegal.
    Switzerland Controlled (Verzeichnis E) Specifically named as a controlled substance under Verzeichnis E since November 1, 2005, pursuant to the Act on the Prohibition of Certain Goods Dangerous to Health.
    Turkey Illegal Classified as a controlled drug. Possession, production, supply, and importation are prohibited under Turkish drug law.
    United Kingdom Class A Controlled as a Class A substance due to its status as an ester of 4-HO-DET, which falls under the tryptamine catch-all clause of the Misuse of Drugs Act 1971. Carries the most severe penalties for possession, production, and supply.
    United States Unscheduled Not federally scheduled under the Controlled Substances Act. However, as a structural analogue of psilocin (4-HO-DMT), which is a Schedule I substance, sale for human consumption or use for illicit purposes could potentially be prosecuted under the Federal Analogue Act.

    Harm Reduction

    drugs.wiki

    4-AcO-DET likely deacetylates in vivo to 4-HO-DET (ethocin), so potency, onset, and duration can vary with metabolism; users report both short (2–4 h) and longer (6–8 h) courses. Anecdotal reports describe stronger, shorter effects via intranasal or smoked routes, but these also carry more irritation and unpredictability; oral is the most characterized and generally lowest risk ROA. Like other 4-substituted tryptamines, nausea and GI unease can occur, particularly on the come-up; fasting 3–4 h and using ginger/antiemetic strategies may help. Avoid mixing with MAOIs, tramadol, DXM, or linezolid due to serotonin toxicity risk; lithium with psychedelics has repeatedly been linked with seizures and severe adverse reactions in community reports. SSRIs/SNRIs and some antipsychotics may attenuate psychedelic effects, but they can still contribute to serotonergic burden; effects can be unpredictable. Misrepresentation in the gray/illicit market is a documented risk (e.g., tryptamines sold as psilocybin or vice versa); reagent testing (Ehrlich for indoles) and lab drug checking reduce this risk, although reagents cannot confirm exact identity. Store away from heat, moisture, and light; 4-AcO esters can hydrolyze over time to 4-HO analogs—color changes (tanning/darkening) have been reported alongside retained potency, but degradation is formulation- and storage-dependent. Tolerance builds rapidly after a single session and decays over about 1–2 weeks; cross-tolerance exists with other classical psychedelics (psilocin/psilocybin, LSD, other 4-sub tryptamines). Set and setting strongly influence outcomes; a trusted sober sitter, safe environment, and clear intentions reduce risk of panic and dangerous behavior. Seek urgent medical help for signs of serotonin toxicity (agitation, hyperthermia, tremor/clonus, confusion), chest pain, persistent vomiting, seizures, or severe confusion; disclose all substances to responders.

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