3,4-Dichloromethylphenidate
Aliases: 3,4-ctmp, 3,4-dcmp, Dichloromethylphenidate, 34ctmp
Categories
Summary
3,4-CTMP is approximately seven times more potent than methylphenidate and has a significantly longer duration of 6-18 hours. A critical safety concern is its agonist activity at 5-HT2B receptors, which can cause pulmonary hypertension and heart valve fibrosis with repeated use. Insufflation is strongly discouraged as the substance has low water solubility, is extremely caustic to nasal tissues, and has poor absorption leading to delayed onset that increases overdose risk. Users must use precise milligram scales due to the extremely low active doses. The very long onset (1-2 hours) and extended duration require careful dose timing to avoid unwanted sleep disruption and accidental overdoses from premature redosing.
Dose Information
| ROA | Light | Common | Strong | Heavy |
|---|---|---|---|---|
| Oral | 2-4mg | 4-6mg | 6-8mg | 8mg+ |
Onset, Duration & After-effects
| ROA | Onset | Peak | Offset | After Effects | Total |
|---|---|---|---|---|---|
| Oral | 1-2 hrs | 3-6 hrs | 4-8 hrs | 2-24 hrs | 240-0 min |
Tolerance
Effects
- Stimulation
- Increased energy/alertness
- Increased Heart Rate
- Vasoconstriction
- Teeth Grinding
- Headaches
- Pupil Dilation
- Temporary Erectile Dysfunction
- Weight loss
- Sweating
- Bruxism
- Headache
- Increased blood pressure
- Abnormal heartbeat
- Stimulant psychosis
- Decreased need for sleep
- Decreased appetite
- Disturbed sleep patterns
- Itchiness
- Spontaneous bodily sensations
- Mouth numbing
- Decreased blood pressure
- Stamina intensification
- Focus Enhancement
- Motivation Enhancement
- Wakefulness
- Analysis Enhancement
- Euphoria
- Increased sociability
- Mood lift
- Cognitive euphoria
- Anxiety
- Aggressiveness
- Emotion suppression
- Dizziness
- Depression
- Paranoia
- Irritability
- Thought deceleration
- Brain zaps
- Cognitive fatigue
- Motivation depression
- Thought Acceleration
- Time Distortion
- Excessive talking
- Moodiness
- Ego inflation
- Thought organization
- Focus intensification
- Visual acuity enhancement
- Increased music appreciation
- Appetite Suppression
- Dehydration
- Double vision
- Disinhibition
- Visual acuity suppression
- Cognitive dysphoria
- Increased sexuality
- Visual and auditory hallucinations
- Drifting
- Optical sliding
- Color tinting
- Tactile intensification